ISSN print edition: 0366-6352 ISSN electronic edition: 1336-9075 Registr. No.: MK SR 9/7 Published monthly

Benzothiazole compounds. IX. Synthesis and comparison of antibacterial activity of esters of (2-benzothiazolyl)acetic acid, (6-X-2-benzothiazolylthio)acetic acid, and of β-(6-X-2-benzothiazolylthio)propionic acid

Ľ. Orosová, V. Sutoris, P. Foltínová, and Š. Haviarová

Drug Research Institute, 801I 00 Bratislava

Abstract:  Alkyl (2-benzothiazolyI)acetates, aryl (6-X-2-benzothiazolylthio)acetates, and alkyl  β-(6-X-2-benzothiazolylthio)propionates (X = H, NO₂, NH₂) were synthesized and tested on some microorganisms. p-Chlorophenyl (2-benzothiazolylthio)acetate (X) and p-nitrophenyl (6-nitro-2-benzothiazolylthio)acetate (XIX) were found to be the most active against nonspecific bacterial flora.

Full paper in Portable Document Format: 302a186.pdf

Chemical Papers 30 (2) 186–194 (1976)